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Results for "

Androgen receptor-IN-2

" in MedChemExpress (MCE) Product Catalog:

6

Inhibitors & Agonists

1

Natural
Products

1

Isotope-Labeled Compounds

Targets Recommended:
Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-136582
    Masofaniten

    Androgen receptor-IN-2

    		 Androgen Receptor Cancer
    Masofaniten (Androgen receptor-IN-2) is a potent and orally active androgen receptor inhibitor. Masofaniten has antitumor activity against prostate cancer .
    Masofaniten
  • HY-13604
    Cyproterone acetate
    2 Publications Verification

    		 Androgen Receptor Endocrinology Cancer
    Cyproterone acetate is an anti-androgen (IC50=7.1 nM) and progestogen synthetic steroid. Cyproterone acetate has affinity with progesteron and with glucocorticoidal receptors .
    Cyproterone acetate
  • HY-W584986
    Androgen receptor degrader-2

    		Androgen Receptor Cancer
    Androgen receptor degrader-2 (compound 9) is a potent androgen receptor degrader. Androgen receptor degrader-2 can be used in research of cancer .
    Androgen receptor degrader-2
  • HY-13604S
    Cyproterone acetate-d3

    		Isotope-Labeled Compounds Androgen Receptor Endocrinology Cancer
    Cyproterone acetate-d3 is deuterium labeled Cyproterone acetate. Cyproterone acetate is an anti-androgen (IC50=7.1 nM) and progestogen synthetic steroid. Cyproterone acetate has affinity with progesteron and with glucocorticoidal receptors[1][2].
    Cyproterone acetate-d3
  • HY-13604R
    Cyproterone acetate (Standard)

    		Androgen Receptor Endocrinology Cancer
    Cyproterone acetate (Standard) is the analytical standard of Cyproterone acetate. This product is intended for research and analytical applications. Cyproterone acetate is an anti-androgen (IC50=7.1 nM) and progestogen synthetic steroid. Cyproterone acetate has affinity with progesteron and with glucocorticoidal receptors .
    Cyproterone acetate (Standard)
  • HY-N7210
    Kahweol acetate

    		Apoptosis Cancer
    Kahweol acetate, a bioactive compound found in coffee, has been identified for its potent anti-cancer properties, particularly in inhibiting the proliferation and migration of prostate cancer cells. Alongside cafestol, it shows dose-dependent effects in suppressing tumor growth and metastasis in both in vitro and in vivo studies. Mechanistically, kahweol acetate and cafestol induce apoptosis, inhibit epithelial-mesenchymal transition, and reduce androgen receptor activity, especially in androgen receptor-positive cells. They also downregulate chemokine receptors CCR2 and CCR5, crucial for cancer progression, without altering their ligand levels. These findings suggest that kahweol acetate, in combination with cafestol, may serve as promising therapeutic agents against prostate cancer .
    Kahweol acetate

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