GPCR Bioassay Screening Services

G protein-coupled receptors (GPCRs) play important roles in cellular physiology and they are popular drug targets for various diseases. About 40% of approved drugs on the market belong to this category. Drug candidate screening and profiling is a critical step in GPCR-centered drug discovery.

MedChemExpress (MCE) can provide high-quality and comprehensive GPCR Bioassay Services. Through efficient, rapid and accurate experimental services, MedChemExpress (MCE) can speed up the discovery and development of new drugs for customers and maximize the benefits of customers.

Key Features

• •Over 100 different GPCR functional cell lines
• •Customized GPCR stable cell line construction
• •High-throughput screening platform: FLIPR PENTA (EMC-CD), BMG PHERAstarFSX, BIOTEK multifunctional plate reader
• •Multiple assay formats including calcium flux, cAMP determination, and Luciferase reporter gene assays
• •Determine drug potency and efficacy in agonist, antagonist, inverse agonist and allosteric modulator modes
• •Stringent QC standards with competitive prices
• •Short turnaround time

The corresponding scheme and price for GPCR Bioassay Screening Services shall be determined after evaluation. For further information on service pricing or technical details, please email sales@MedChemExpress.com or contact MedChemExpress (MCE) sales staff directly.