2. GPCR/G Protein
  3. Adenosine Receptor
  4. A3AR antagonist 2

A3AR antagonist 2 (compound 18) is a potent Human A3 adenosine receptor antagonist with an Ki value of 4.54 nM.

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A3AR antagonist 2 Chemical Structure

A3AR antagonist 2 Chemical Structure

CAS No. : 1144161-05-6

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A3AR antagonist 2 Related Antibodies

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Description

A3AR antagonist 2 (compound 18) is a potent Human A3 adenosine receptor antagonist with an Ki value of 4.54 nM[1].

IC50 & Target[1]

hA3

4.54 nM (Ki)

Molecular Weight

412.40

Formula

C22H16N6O3
CAS No.
SMILES

O=C(NC1=NC2=NC=CC=C2N3C1=NN(C4=CC=C(OC)C=C4)C3=O)C5=CC=CC=C5
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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A3AR antagonist 2 Related Classifications

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    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

A3AR antagonist 21144161-05-6Adenosine ReceptorP1 receptorInhibitorinhibitorinhibit

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