2. Vitamin D Related/Nuclear Receptor
  3. Estrogen Receptor/ERR
  4. 4'-Raloxifene-β-D-glucopyranoside

4'-Raloxifene-β-D-glucopyranoside, a metabolite of Raloxifene, is a benzothiophene glucuronidated at the 4' postion. 4'-Raloxifene-β-D-glucopyranoside is a selective and orally active estrogen receptor antagonist. 4'-Raloxifene-β-D-glucopyranoside can be used for inhibiting bone loss and resorption, and lowering lipid levels. 4'-Raloxifene-β-D-glucopyranoside, example 5, is extracted from patent US5567820A.

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4'-Raloxifene-β-D-glucopyranoside Chemical Structure

4'-Raloxifene-β-D-glucopyranoside Chemical Structure

CAS No. : 334758-19-9

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4'-Raloxifene-β-D-glucopyranoside Related Antibodies

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Estrogen receptor ERα ERβ ERRα ERRβ ERRγ

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Description

4'-Raloxifene-β-D-glucopyranoside, a metabolite of Raloxifene, is a benzothiophene glucuronidated at the 4' postion. 4'-Raloxifene-β-D-glucopyranoside is a selective and orally active estrogen receptor antagonist. 4'-Raloxifene-β-D-glucopyranoside can be used for inhibiting bone loss and resorption, and lowering lipid levels. 4'-Raloxifene-β-D-glucopyranoside, example 5, is extracted from patent US5567820A[1].

IC50 & Target

IC50: estrogen receptor[1]
Molecular Weight

635.72

Formula

C34H37NO9S
CAS No.
SMILES

O=C(C1=C(C2=CC=C(O[C@H]3[C@@H]([C@H]([C@@H]([C@@H](CO)O3)O)O)O)C=C2)SC4=CC(O)=CC=C41)C5=CC=C(OCCN6CCCCC6)C=C5
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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4'-Raloxifene-β-D-glucopyranoside Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

4'-Raloxifene-β-D-glucopyranoside334758-19-9Estrogen Receptor/ERRmetabolitebone lossbone resorption lower lipid RaloxifeneInhibitorinhibitorinhibit

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