2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. 5-HT6R antagonist 6

5-HT6R antagonist 6 exhibits high affinity and selectivity for 5-HT6R , with a Ki value of 42 nM. 5-HT6R antagonist 6 shows weak antiproliferative activity against tumor cells and low toxicity to normal cells. 5-HT6R antagonist 6 can be used in the study of cancer.

For research use only. We do not sell to patients.

5-HT6R antagonist 6 Chemical Structure

5-HT6R antagonist 6 Chemical Structure

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Description

5-HT6R antagonist 6 exhibits high affinity and selectivity for 5-HT6R , with a Ki value of 42 nM. 5-HT6R antagonist 6 shows weak antiproliferative activity against tumor cells and low toxicity to normal cells. 5-HT6R antagonist 6 can be used in the study of cancer[1].

IC50 & Target[1]

5-HT6 Receptor

42 nM (Ki)

Molecular Weight

434.55

Formula

C24H26N4O2S
SMILES

O=S(C1=C2C=CC=CC2=CC=C1)(NCCCCCCNC3=NC=C4C=CC=CC4=N3)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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5-HT6R antagonist 6 Related Classifications

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Keywords:

5-HT6R antagonist 65-HT ReceptorSerotonin Receptor5-hydroxytryptamine Receptor1321N1U87MGU-251LN-229MCF7AsPC-1NHAInhibitorinhibitorinhibit

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5-HT6R antagonist 6
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