2. Signaling Pathways
  3. GPCR/G Protein
  4. RXFP Receptor
  5. RXFP Receptor Antagonist

RXFP Receptor Antagonist

RXFP Receptor Antagonist (1):

Cat. No. Product Name Effect Purity
  • HY-162401
    AZ7976
    		Antagonist
    AZ7976 (Compound 42) is a highly selective agonist for the Relaxin Family Peptide Receptor 1 (RXFP1) (pEC50 > 10.5). AZ7976 enhances RXFP1's cAMP signaling through an allosteric mechanism, thereby physiologically increasing heart rate. AZ7976 can be used in the field of cardiovascular disease research.