2. GPCR/G Protein
  3. Adenosine Receptor
  4. Adenosine receptor antagonist 1

Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aR than A2bR.

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Adenosine receptor antagonist 1 Chemical Structure

Adenosine receptor antagonist 1 Chemical Structure

CAS No. : 2682930-40-9

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Adenosine receptor antagonist 1 Related Antibodies

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Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

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Description

Adenosine receptor antagonist 1 is a A2aR-selective antagonist with an IC50 of 0.29 nM and displays 14-fold more selective for A2aR than A2bR.

IC50 & Target

A2AR

0.29 nM (IC50)

Molecular Weight

447.85

Formula

C22H15ClFN7O
CAS No.
SMILES

NC1=NC(C2=CC=CC=C2)=C(C3=NC(CC4=C(C=C(C=N4)F)Cl)=NN13)C5=CNC(C=C5)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Adenosine receptor antagonist 1 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Adenosine receptor antagonist 12682930-40-9Adenosine receptor antagonist1Adenosine receptor antagonist-1Adenosine ReceptorP1 receptorInhibitorinhibitorinhibit

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