2. Epigenetics
  3. Epigenetic Reader Domain
  4. BET BD2-IN-3

BET BD2-IN-3 (compound I-58) is an inhibitor of BET, targeting the BD2 domain of BET. BET BD2-IN-3 can be radiolabeled with [11C] for positron emission tomography (PET) imaging. BET [11C]BD2-IN-3 showed suitable biodistribution in peripheral organs and tissues in PET applications in mice.

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BET BD2-IN-3 Chemical Structure

BET BD2-IN-3 Chemical Structure

CAS No. : 2677039-66-4

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BET BD2-IN-3 Related Antibodies

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Description

BET BD2-IN-3 (compound I-58) is an inhibitor of BET, targeting the BD2 domain of BET. BET BD2-IN-3 can be radiolabeled with [11C] for positron emission tomography (PET) imaging. BET [11C]BD2-IN-3 showed suitable biodistribution in peripheral organs and tissues in PET applications in mice[1].

IC50 & Target

BET BD2[1]
Molecular Weight

450.57

Formula

C29H30N4O
CAS No.
SMILES

O=C1N(C)C2=CC3=CC=CC=C3N(CC4=CC=CC(NC5CCN(C)CC5)=C4)C6=CC=CC1=C26
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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BET BD2-IN-3 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

BET BD2-IN-32677039-66-4Epigenetic Reader DomainInhibitorinhibitorinhibit

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