2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. GABA Receptor
  4. CGP 54626 hydrochloride

CGP 54626 (hydrochloride) is a selective antagonist of GABAB receptor with an IC50 value of 4 nM. CGP 54626 (hydrochloride) can be used to investigate the role of GABAB receptors in neurological signaling.

For research use only. We do not sell to patients.

CGP 54626 hydrochloride Chemical Structure

CGP 54626 hydrochloride Chemical Structure

CAS No. : 149184-21-4

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Based on 1 publication(s) in Google Scholar

Other Forms of CGP 54626 hydrochloride:

CGP 54626 hydrochloride Related Antibodies

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1 Publications Citing Use of MCE CGP 54626 hydrochloride

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Description

CGP 54626 (hydrochloride) is a selective antagonist of GABAB receptor with an IC50 value of 4 nM. CGP 54626 (hydrochloride) can be used to investigate the role of GABAB receptors in neurological signaling[1].

Cellular Effect
Cell Line Type Value Description References
CHO IC50
6.4 nM
Compound: CGP-54626
Displacement of [3H]CGP54626 from human recombinant GABAB1A receptor expressed in CHO cells after 3 hrs
Displacement of [3H]CGP54626 from human recombinant GABAB1A receptor expressed in CHO cells after 3 hrs
[PMID: 23403082]
Molecular Weight

444.76

Formula

C18H29Cl3NO3P
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=P(C[C@@H](O)CN[C@H](C1=CC=C(Cl)C(Cl)=C1)C)(CC2CCCCC2)O.Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, protect from light, stored under nitrogen

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen)

Purity & Documentation
References
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CGP 54626 hydrochloride Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CGP 54626149184-21-4CGP54626CGP-54626GABA ReceptorGamma-aminobutyric acid Receptorγ-Aminobutyric acid ReceptorInhibitorinhibitorinhibit

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CGP 54626 hydrochloride
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HY-101378
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