Darifenacin (hydrobromide) (Standard) (Synonyms: UK-88525 (hydrobromide) (Standard))

Cat. No.: HY-A0012R Purity: ≥98%: FAQs
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Darifenacin (hydrobromide) (Standard) is the analytical standard of Darifenacin (hydrobromide). This product is intended for research and analytical applications. Darifenacin (hydrobromide) is a selective and orally active M3 muscarinic receptor (M3R) antagonist with a pKi of 8.9. Darifenacin (hydrobromide) binds >20-fold more specifically to M3R than to other muscarinic receptors. Darifenacin (hydrobromide) can be used in the study of urinary incontinence and other symptoms of overactive bladder. Darifenacin (hydrobromide) inhibits tumor growth in colorectal cancer cells and has anti-tumor effects.

For research use only. We do not sell to patients.

Darifenacin (hydrobromide) (Standard) Chemical Structure

CAS No. : 133099-07-7

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Description	Darifenacin (hydrobromide) (Standard) is the analytical standard of Darifenacin (hydrobromide). This product is intended for research and analytical applications. Darifenacin (hydrobromide) is a selective and orally active M3 muscarinic receptor (M3R) antagonist with a pKi of 8.9. Darifenacin (hydrobromide) binds >20-fold more specifically to M3R than to other muscarinic receptors. Darifenacin (hydrobromide) can be used in the study of urinary incontinence and other symptoms of overactive bladder. Darifenacin (hydrobromide) inhibits tumor growth in colorectal cancer cells and has anti-tumor effects.
Molecular Weight	507.46
Formula	C₂₈H₃₁BrN₂O₂
CAS No.	133099-07-7
SMILES	O=C(C(C1=CC=CC=C1)([C@@H]2CCN(CCC3=CC4=C(OCC4)C=C3)C2)C5=CC=CC=C5)N.Br
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation	Handling Instructions (2659 KB)

Darifenacin (hydrobromide) (Standard) Related Classifications

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass		Concentration		Volume		Molecular Weight *
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The dilution calculator equation

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Darifenacin (hydrobromide) (Standard)133099-07-7UK-88525 hydrobromide (Standard)mAChRp38 MAPKAktMuscarinic acetylcholine receptorPKBProtein kinase BLiver damage modelColorectal cancer modelHT-29 cellsSW480 cellsCoronary arterial smooth muscle cellsM3 Muscarinic Receptor AntagonistInhibitorinhibitorinhibit

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Darifenacin (hydrobromide) (Standard) (Synonyms: UK-88525 (hydrobromide) (Standard))

Product Information

Purity & Documentation

Customer Review

Darifenacin (hydrobromide) (Standard) Related Classifications

Molarity Calculator

Dilution Calculator