DG013A formate

Cat. No.: HY-139907B Purity: 99.60%: FAQs
Data Sheet SDS COA Handling Instructions Technical Support

DG013A (formate) is a phosphinic acid tripeptide mimetic inhibitor. DG013A (formate) displays significantly weak affinity for both ERAP1 (IC₅₀=33 nM) and ERAP2 (IC₅₀=11 nM). DG013A (formate) can be used for the research of autoimmune disease and cancer.

For research use only. We do not sell to patients.

DG013A formate Chemical Structure

Size	Stock	Quantity
1 mg	In-stock	Estimated Time of Arrival: December 31
5 mg	In-stock	Estimated Time of Arrival: December 31
10 mg	In-stock	Estimated Time of Arrival: December 31
25 mg	In-stock	Estimated Time of Arrival: December 31
50 mg	Get quote
100 mg	Get quote

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This product is a controlled substance and not for sale in your territory.

Other Forms of DG013A formate:

DG013B Get quote
DG013B formate Get quote
DG013A Get quote

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Biological Activity
Purity & Documentation
References
Customer Review

Description

Molecular Weight

530.99

Formula

C₂₇H₃₇N₄O₄P.2/5CH₂O₂

Appearance

Solid

Color

White to off-white

SMILES

O=P([C@@H](N)CCC1=CC=CC=C1)(O)C[C@@H](CC(C)C)C(N[C@H](C(N)=O)CC2=CNC3=CC=CC=C23)=O.O=CO.[0.4]

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
In solvent	-80°C	6 months
	-20°C	1 month

Purity & Documentation

Purity: 99.60%

Select Batch:

Data Sheet (270 KB) SDS (251 KB)

COA (254 KB) HNMR (287 KB) LCMS (100 KB)

Handling Instructions (2659 KB)

References

[1]. Birgit Wilding, et al. Investigating the phosphinic acid tripeptide mimetic DG013A as a tool compound inhibitor of the M1-aminopeptidase ERAP1. Bioorg Med Chem Lett. 2021 Jun 15;42:128050. [Content Brief]

DG013A formate Related Classifications

Molarity Calculator
Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass		Concentration		Volume		Molecular Weight *
	=		×		×

The dilution calculator equation

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

DG013A formateAminopeptidaseautoimmune diseasecancerERAP1Chemical probeM1-aminopeptidasePermeabilityInhibitorinhibitorinhibit

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