2. Others Vitamin D Related/Nuclear Receptor
  3. Isotope-Labeled Compounds Estrogen Receptor/ERR
  4. Elacestrant-d4-1

Elacestrant-d4-1 is the deuterium labeled Elacestrant (HY-19822). Elacestrant is an orally available and selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.

For research use only. We do not sell to patients.

Elacestrant-d<sub>4</sub>-1 Chemical Structure

Elacestrant-d4-1 Chemical Structure

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Other Forms of Elacestrant-d4-1:

Elacestrant-d4-1 Related Antibodies

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Estrogen receptor ERα ERβ ERRα ERRβ ERRγ

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Description

Elacestrant-d4-1 is the deuterium labeled Elacestrant (HY-19822). Elacestrant is an orally available and selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively[1][2].

Molecular Weight

462.66

Formula

C30H34D4N2O2
Unlabeled CAS

722533-56-4
SMILES

OC1=C([2H])C=C2C[C@H](C3=CC([2H])=C(OC)C([2H])=C3N(CC)CC4=CC=C(CCNCC)C=C4)CCC2=C1[2H]
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Elacestrant-d4-1 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Elacestrant-d4-1RAD1901-d4-1Isotope-Labeled CompoundsEstrogen Receptor/ERRInhibitorinhibitorinhibit

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