2. Membrane Transporter/Ion Channel
  3. OAT URAT1
  4. Epaminurad hydrochloride

Epaminurad hydrochloride  (Synonyms: UR-1102 hydrochloride; URC-102 hydrochloride)

Cat. No.: HY-111345A
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Epaminurad (UR-1102) hydrochloride is an orally active, potent and selective URAT1 (urate transporter 1) inhibitor, with a Ki of 0.057 μM. Epaminurad hydrochloride quite modestly inhibits OAT1 and OAT3 (organic anion transporter). Epaminurad hydrochloride is a uricosuric agent. Epaminurad hydrochloride can be used for gout and hyperuricemia research.

For research use only. We do not sell to patients.

Epaminurad hydrochloride Chemical Structure

Epaminurad hydrochloride Chemical Structure

CAS No. : 1198153-46-6

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Epaminurad hydrochloride Related Antibodies

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Description

Epaminurad (UR-1102) hydrochloride is an orally active, potent and selective URAT1 (urate transporter 1) inhibitor, with a Ki of 0.057 μM. Epaminurad hydrochloride quite modestly inhibits OAT1 and OAT3 (organic anion transporter). Epaminurad hydrochloride is a uricosuric agent. Epaminurad hydrochloride can be used for gout and hyperuricemia research[1].

IC50 & Target

Ki: 0.057 ± 0.036 μM (URAT1), 2.4 ± 0.2 μM (OAT3), 7.2 ± 0.8 μM (OAT1)[1].
Molecular Weight

450.51

Formula

C14H11Br2ClN2O3
CAS No.
SMILES

O=C(N1C2=C(OCC1)C=CN=C2)C3=CC(Br)=C(C(Br)=C3)O.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Epaminurad hydrochloride Related Classifications

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Epaminurad1198153-46-6UR-1102URC-102UR1102UR 1102URC102URC 102OATURAT1Organic anion transporterUrate transporter 1SLC22A12HEK293 cellsUricosuricgouthyperuricemiap-aminohippuric acidurateInhibitorinhibitorinhibit

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