2. MAPK/ERK Pathway Stem Cell/Wnt
  3. ERK
  4. ERK2 allosteric-IN-1

ERK2 allosteric-IN-1 (compound 1) is a selective and allosteric ERK2 inhibitor with the IC50 of 11 μM.

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ERK2 allosteric-IN-1 Chemical Structure

ERK2 allosteric-IN-1 Chemical Structure

CAS No. : 872591-16-7

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ERK2 allosteric-IN-1 Related Antibodies

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Description

ERK2 allosteric-IN-1 (compound 1) is a selective and allosteric ERK2 inhibitor with the IC50 of 11 μM[1].

IC50 & Target

ERK2

11 μM (IC50)

Molecular Weight

432.43

Formula

C22H20N6O4
CAS No.
SMILES

O=C(CN1C=NC(N(C2=CC(C)=C(C)C=C2)N=N3)=C3C1=O)NCC4=CC5=C(OCO5)C=C4
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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ERK2 allosteric-IN-1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

ERK2 allosteric-IN-1872591-16-7ERKExtracellular signal regulated kinasesCancerERK2type 2 diabeteInhibitorinhibitorinhibit

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