Fluphenazine enanthate

Cat. No.: HY-107947: FAQs
Data Sheet Handling Instructions

Molarity Calculator

Fluphenazine enanthate is the first long-acting injectable (LAI) antipsychotic for the treatment of schizophrenia.

For research use only. We do not sell to patients.

Fluphenazine enanthate Chemical Structure

CAS No. : 2746-81-8

Size		Stock
MOQ		Minimum order quantity
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote
Other size		Get quote

Synthetic products have potential research and development risk.

* Please select Quantity before adding items.

This product is a controlled substance and not for sale in your territory.

Featured Recommendations

•Related Small Molecules:

•Related Proteins:

Biological Activity
Purity & Documentation
References
Customer Review

Description

Fluphenazine enanthate is the first long-acting injectable (LAI) antipsychotic for the treatment of schizophrenia^[1]^[2].

In Vivo

Fluphenazine enanthate (2,4, 8 mg/kg; IM) significant inhibition of the avoidance performance is observed as long as 16, 23, and 28 days, respectively^[1].
Fluphenazine enanthate (8 mg/kg) drinking behavior is almost completely suppressed for 24 hours immediately following the administration^[1].
Fluphenazine enanthate (8 mg/kg) produces transient body weight Iosses in the rats^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model:	Fifty-four male adult rats of Wistar strain^[1]
Dosage:	2, 4, and 8 mg/kg
Administration:	Index medicus (IM )
Result:	Three doses of Fluphenazine enanthate significant inhibition of the avoidance performance was observed as long as 16, 23, and 28 days, respectively.

Molecular Weight

549.69

Formula

C₂₉H₃₈F₃N₃O₂S

CAS No.

2746-81-8

SMILES

CCCCCCC(OCCN1CCN(CCCN2C3=C(C=CC=C3)SC4=CC=C(C(F)(F)F)C=C24)CC1)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Kuribara H, et al. Effects of fluphenazine enanthate and fluphenazine decanoate on discriminated avoidanceresponse and water drinking behavior in rats. Psychopharmacology (Berl). 1979 Sep;65(1):1-6. [Content Brief]

[2]. Brissos S, et al. The role of long-acting injectable antipsychotics in schizophrenia: a critical appraisal. Ther Adv Psychopharmacol. 2014 Oct;4(5):198-219. [Content Brief]