2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. Proxyfan Oxalate

Proxyfan Oxalate is a potent histamine H3 receptor antagonist with Ki values of 2.9 nM and 2.7 nM for rat and human H3 receptor, respectively. Proxyfan Oxalate is over 1000-fold more potent at H3 receptors than other histamine receptors.

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Proxyfan Oxalate Chemical Structure

Proxyfan Oxalate Chemical Structure

CAS No. : 1620017-81-3

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Other Forms of Proxyfan Oxalate:

Proxyfan Oxalate Related Antibodies

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Description

Proxyfan Oxalate is a potent histamine H3 receptor antagonist with Ki values of 2.9 nM and 2.7 nM for rat and human H3 receptor, respectively. Proxyfan Oxalate is over 1000-fold more potent at H3 receptors than other histamine receptors[1][2].

IC50 & Target[1]

Rat H3LR

2.9 nM (Ki)

Human H3LR

2.7 nM (Ki)

Molecular Weight

306.31

Formula

C15H18N2O5
CAS No.
SMILES

O=C(O)C(O)=O.C1(CCCOCC2=CC=CC=C2)=CNC=N1
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Proxyfan Oxalate Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Proxyfan1620017-81-3Histamine Receptorhistamine H3 receptorneutral antagonistInhibitorinhibitorinhibit

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HY-107557A
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