1. Vitamin D Related/Nuclear Receptor Apoptosis Metabolic Enzyme/Protease Immunology/Inflammation NF-κB
  2. Estrogen Receptor/ERR Apoptosis Reactive Oxygen Species
  3. rel-Levormeloxifene

rel-Levormeloxifene  (Synonyms: rel-L-Centchroman; Ormeloxifene)

Cat. No.: HY-122359A
Handling Instructions

rel-Levormeloxifene (rel-L-Centchroman) is the relative configuration of Levormeloxifene (HY-122359). rel-Levormeloxifene is a selective estrogen receptor modulator (SERM). rel-Levormeloxifene inhibits proliferation of leukemia cells with IC50 about 7 μM, arrests cell cycle at G0/G1 phase, and induces apoptosis. rel-Levormeloxifene induces differentation of myelogenesis leukemia, and enhances ROS production in K562 cells.

For research use only. We do not sell to patients.

rel-Levormeloxifene Chemical Structure

rel-Levormeloxifene Chemical Structure

CAS No. : 31477-60-8

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Description

rel-Levormeloxifene (rel-L-Centchroman) is the relative configuration of Levormeloxifene (HY-122359). rel-Levormeloxifene is a selective estrogen receptor modulator (SERM). rel-Levormeloxifene inhibits proliferation of leukemia cells with IC50 about 7 μM, arrests cell cycle at G0/G1 phase, and induces apoptosis. rel-Levormeloxifene induces differentation of myelogenesis leukemia, and enhances ROS production in K562 cells[1].

Molecular Weight

457.60

Formula

C30H35NO3

CAS No.
SMILES

CC1(C)[C@@H](C2=CC=CC=C2)[C@H](C3=CC=C(OCCN4CCCC4)C=C3)C5=CC=C(OC)C=C5O1

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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rel-Levormeloxifene
Cat. No.:
HY-122359A
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