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Results for "

BRD4 degrader-5

" in MedChemExpress (MCE) Product Catalog:

5

Inhibitors & Agonists

1

Click Chemistry

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-133737
    PROTAC BRD4 Degrader-5

    		PROTACs Epigenetic Reader Domain Cancer
    PROTAC BRD4 Degrader-5 is a PROTAC connected by ligands for von Hippel-Lindau and BRD4. PROTAC BRD4 Degrader-5 can potent degrade BRD4 in HER2 positive and negative breast cancer cell lines .
    PROTAC BRD4 Degrader-5
  • HY-133736
    PROTAC BRD4 Degrader-5-CO-PEG3-N3

    		PROTAC-Linker Conjugates for PAC ADC Cytotoxin Cancer
    PROTAC BRD4 Degrader-5-CO-PEG3-N3 (Compound 2) is a PROTAC-linker Conjugate for PAC, comprises the BRD4 degrader GNE-987 and PEG-based linker . PROTAC BRD4 Degrader-5-CO-PEG3-N3 is a click chemistry reagent, it contains an Azide group and can undergo copper-catalyzed azide-alkyne cycloaddition reaction (CuAAc) with molecules containing Alkyne groups. It can also undergo strain-promoted alkyne-azide cycloaddition (SPAAC) reactions with molecules containing DBCO or BCN groups.
    PROTAC BRD4 Degrader-5-CO-PEG3-N3
  • HY-131387
    (S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2

    		E3 Ligase Ligand-Linker Conjugates Cancer
    (S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2 is a synthesized E3 ligase ligand-linker conjugate that incorporates the a VHL ligand and a linker. (S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2 can be used in PROTAC BRD4 Degrader-5 (HY-133737) and PROTAC BRD4 Degrader-5-CO-PEG3-N3 (HY-133736) .
    (S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2
  • HY-170989
    BRD4 degrader-5

    		AUTACs Epigenetic Reader Domain Autophagy Cancer
    BRD4 degrader-5 (Compound 23) is a hydrophobic tag (HyTag)-based protein degrader for BRD4 (DC50 = 24.7 μM) through ER stress and autophagy-lysosome pathway. BRD4 degrader-5 inhibits the proliferation of cancer cell 4T1 with an IC50 of 20.6 μM .
    BRD4 degrader-5
  • HY-160694
    cBu-Cit-PROTAC BRD4 Degrader-5

    		PROTACs Cancer
    cBu-Cit-PROTAC BRD4 Degrader-5 is a PROTAC that degrades BRD4 by association with cBu-Cit. cBu-Cit-PROTAC BRD4 Degrader-5 can effectively inhibit BRD4 in HER2 positive and negative breast cancer cell lines. cBu-Cit-PROTAC BRD4 Degrader-5 has a single bond and can be conjugated to an ADC antibody to form a PAC .
    cBu-Cit-PROTAC BRD4 Degrader-5

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