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Urotensin-II receptor antagonist-1

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Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-10672
    Urotensin-II receptor antagonist-1

    		Urotensin Receptor Cardiovascular Disease
    Urotensin-II receptor antagonist-1 (compound 1) is a selective human Urotensin II receptor antagonist with low oral bioavailability (F=0-3%, rat) and Ki=16 nM (HEK293 cells expressing human recombinant UT receptor). Urotensin-II receptor antagonist-1 inhibits cytochrome P450 (IC50=0.75 μM, CYP2D6; 1.4 μM, CYP3A4), inhibits kappa opioid receptors (EC50=3.2 μM), and targets cardiac sodium channels (Ki=2.5 μM).
    Urotensin-II receptor antagonist-1

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