2. GPCR/G Protein Neuronal Signaling Anti-infection
  3. 5-HT Receptor Bacterial
  4. Trimipramine maleate (Standard)

Trimipramine maleate (Standard) 

Cat. No.: HY-B1213R Purity: ≥98%
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Trimipramine (maleate) (Standard) is the analytical standard of Trimipramine (maleate). This product is intended for research and analytical applications. Trimipramine maleate is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively. Trimipramine maleate is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 μM, 2.11 μM, 3.72 μM, 8.00 μM, respectively. Trimipramine maleate has vascular activity and anxiolytic efficacy.

For research use only. We do not sell to patients.

Trimipramine maleate (Standard) Chemical Structure

Trimipramine maleate (Standard) Chemical Structure

CAS No. : 521-78-8

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Description

Trimipramine (maleate) (Standard) is the analytical standard of Trimipramine (maleate). This product is intended for research and analytical applications. Trimipramine maleate is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively. Trimipramine maleate is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 μM, 2.11 μM, 3.72 μM, 8.00 μM, respectively. Trimipramine maleate has vascular activity and anxiolytic efficacy.

Molecular Weight

410.51

Formula

C24H30N2O4
CAS No.
SMILES

CC(CN(C)C)CN1C2=C(C=CC=C2)CCC3=C1C=CC=C3.O=C(O)/C=C\C(O)=O
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
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Trimipramine maleate (Standard) Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Trimipramine maleate (Standard)521-78-85-HT ReceptorBacterialSerotonin Receptor5-hydroxytryptamine Receptorantidepressants5-HT5-hydroxytryptamineserotonin5-HTlc receptors5-HTIA receptorsdopamineDADA D2 receptor5-HT1C5-HT25-HT1Aanxiolyticneurological diseasenoradrenalinehNAThSERThDAThuman organic cation transportershOCT1hOCT2hOCT3Inhibitorinhibitorinhibit

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