2. GPCR/G Protein Neuronal Signaling
  3. mAChR
  4. VU6016235

VU6016235 is a highly selective, orally available, positive allosteric modulator of the M4 mAChR with in vivo inhibitory potency in animal models of psychosis..

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VU6016235 Chemical Structure

VU6016235 Chemical Structure

CAS No. : 2344787-70-6

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VU6016235 Related Antibodies

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Description

VU6016235 is a highly selective, orally available, positive allosteric modulator of the M4 mAChR with in vivo inhibitory potency in animal models of psychosis.[1].

Molecular Weight

378.49

Formula

C21H22N4OS
CAS No.
SMILES

CC1=NC2=C(C3=C(S2)C(NCC4=CC=C(C=C4)C(C)(O)C)=NC=C3)C(C)=N1
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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VU6016235 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

VU60162352344787-70-6VU 6016235VU-6016235mAChRMuscarinic acetylcholine receptorInhibitorinhibitorinhibit

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HY-169178
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