2. GPCR/G Protein
  3. Mas-related G-protein-coupled Receptor (MRGPR)
  4. (4′R)-TGR5 Receptor Agonist 4

(4′R)-TGR5 Receptor Agonist 4 is the R enantiomer of TGR5 Receptor Agonist 4 (HY-156830). TGR5 Receptor Agonist 4 is an agonist of Bile Acid Receptor (TGR5), with EC50 for hTGR5 and mTGR5 of 2 nM and 3 nM, respectively. TGR5 Receptor Agonist 4 plays important roles in hypoglycemic and weight loss.

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(4′R)-TGR5 Receptor Agonist 4 Chemical Structure

(4′R)-TGR5 Receptor Agonist 4 Chemical Structure

CAS No. : 1872436-55-9

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Other Forms of (4′R)-TGR5 Receptor Agonist 4:

(4′R)-TGR5 Receptor Agonist 4 Related Antibodies

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Description

(4′R)-TGR5 Receptor Agonist 4 is the R enantiomer of TGR5 Receptor Agonist 4 (HY-156830). TGR5 Receptor Agonist 4 is an agonist of Bile Acid Receptor (TGR5), with EC50 for hTGR5 and mTGR5 of 2 nM and 3 nM, respectively. TGR5 Receptor Agonist 4 plays important roles in hypoglycemic and weight loss[1].

Molecular Weight

470.95

Formula

C25H27ClN2O5
CAS No.
SMILES

COC(C=CC=C1)=C1COC(C([C@@H](C2=CN=C(Cl)C=C2)C3)=C(C)N(C[C@H]4CCCO4)C3=O)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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(4′R)-TGR5 Receptor Agonist 4 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

(4′R)-TGR5 Receptor Agonist 41872436-55-9Mas-related G-protein-coupled Receptor (MRGPR)hypoglycemic and weight lossInhibitorinhibitorinhibit

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