2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. 5-HT2A/5-HT2C inverse agonist 1

5-HT2A/5-HT2C inverse agonist 1 is a potent and dual 5-HT2A and 5-HT2C receptor inverse agonist with a hERG inhibitions, thus avoiding cardiovascular risks. 5-HT2A/5-HT2C inverse agonist 1 shows significant antipsychotic efficacy in the MK-801 (HY-15084B)-induced mouse model. 5-HT2A/5-HT2C inverse agonist 1 is promising for research of psychosis.

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5-HT2A/5-HT2C inverse agonist 1 Chemical Structure

5-HT2A/5-HT2C inverse agonist 1 Chemical Structure

CAS No. : 2718990-76-0

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5-HT2A/5-HT2C inverse agonist 1 Related Antibodies

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Description

5-HT2A/5-HT2C inverse agonist 1 is a potent and dual 5-HT2A and 5-HT2C receptor inverse agonist with a hERG inhibitions, thus avoiding cardiovascular risks. 5-HT2A/5-HT2C inverse agonist 1 shows significant antipsychotic efficacy in the MK-801 (HY-15084B)-induced mouse model. 5-HT2A/5-HT2C inverse agonist 1 is promising for research of psychosis[1].

Molecular Weight

425.57

Formula

C24H35N5O2
CAS No.
SMILES

CN(C=C1)N=C1CN([C@@H]2C3(CN(CC2)C)CC3)C(NCC4=CC=C(C=C4)OCCC)=O
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Room temperature in continental US; may vary elsewhere.
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Purity & Documentation
References
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5-HT2A/5-HT2C inverse agonist 1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

5-HT2A/5-HT2C inverse agonist 12718990-76-05-HT ReceptorSerotonin Receptor5-hydroxytryptamine Receptor5-HT2A receptor5-HT2C receptorhERGcardiovascular risksantipsychotic efficacymousepsychosisInhibitorinhibitorinhibit

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