1. GPCR/G Protein Neuronal Signaling
  2. 5-HT Receptor
  3. 5-HT2A/5-HT2C inverse agonist 1

5-HT2A/5-HT2C inverse agonist 1 is a potent and dual 5-HT2A and 5-HT2C receptor inverse agonist with a hERG inhibitions, thus avoiding cardiovascular risks. 5-HT2A/5-HT2C inverse agonist 1 shows significant antipsychotic efficacy in the MK-801 (HY-15084B)-induced mouse model. 5-HT2A/5-HT2C inverse agonist 1 is promising for research of psychosis.

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5-HT2A/5-HT2C inverse agonist 1 Chemical Structure

5-HT2A/5-HT2C inverse agonist 1 Chemical Structure

CAS No. : 2718990-76-0

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Description

5-HT2A/5-HT2C inverse agonist 1 is a potent and dual 5-HT2A and 5-HT2C receptor inverse agonist with a hERG inhibitions, thus avoiding cardiovascular risks. 5-HT2A/5-HT2C inverse agonist 1 shows significant antipsychotic efficacy in the MK-801 (HY-15084B)-induced mouse model. 5-HT2A/5-HT2C inverse agonist 1 is promising for research of psychosis[1].

Molecular Weight

425.57

Formula

C24H35N5O2

CAS No.
SMILES

CN(C=C1)N=C1CN([C@@H]2C3(CN(CC2)C)CC3)C(NCC4=CC=C(C=C4)OCCC)=O

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5-HT2A/5-HT2C inverse agonist 1 Related Classifications

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5-HT2A/5-HT2C inverse agonist 1
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HY-169001
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