1. GPCR/G Protein Neuronal Signaling
  2. 5-HT Receptor
  3. 5-HT2A antagonist 3

5-HT2A antagonist 3 (Formula (III)) is a 5-HT2A receptor antagonist and inverse agonist with a pIC50 of 8.7 and a pKi of 9. 5-HT2A antagonist 3 can be utilized in neurological reesearch.

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5-HT2A antagonist 3 Chemical Structure

5-HT2A antagonist 3 Chemical Structure

CAS No. : 1134815-69-2

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Description

5-HT2A antagonist 3 (Formula (III)) is a 5-HT2A receptor antagonist and inverse agonist with a pIC50 of 8.7 and a pKi of 9. 5-HT2A antagonist 3 can be utilized in neurological reesearch[1].

IC50 & Target

5-HT2A Receptor

9 (pKi)

Molecular Weight

443.55

Formula

C25H34FN3O3

CAS No.
SMILES

O=C(N(C1CCN(CC1)C)CC2=CC=C(C=C2)F)NCC3=CC=C(C=C3)OCC(C)(C)O

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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5-HT2A antagonist 3 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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5-HT2A antagonist 3
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HY-171235
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