5-Hydroxymethyl tolterodine formate (Synonyms: PNU-200577 formic)

Cat. No.: HY-76569B: FAQs
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5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine (HY-A0024) and Fesoterodine (HY-70053). 5-Hydroxymethyl tolterodine (formate) is formed from tolterodine by the cytochrome P450 (CYP) isoform CYP2D6 and from fesoterodine by plasma esterases.

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5-Hydroxymethyl tolterodine formate Chemical Structure

CAS No. : 380636-49-7

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Other In-stock Forms of 5-Hydroxymethyl tolterodine formate:

Desfesoterodine

Other Forms of 5-Hydroxymethyl tolterodine formate:

Desfesoterodine In-stock
(R)-Hydroxytolterodine-d₁₄ Get quote

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Description	5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine (HY-A0024) and Fesoterodine (HY-70053). 5-Hydroxymethyl tolterodine (formate) is formed from tolterodine by the cytochrome P450 (CYP) isoform CYP2D6 and from fesoterodine by plasma esterases.
Molecular Weight	387.51
Formula	C₂₃H₃₃NO₄
CAS No.	380636-49-7
SMILES	OC1=C(C=C(CO)C=C1)[C@@H](C2=CC=CC=C2)CCN(C(C)C)C(C)C.OC=O
Shipping	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation	Data Sheet (268 KB) Handling Instructions (2659 KB)
References	[1]. L Nilvebrant, et al. Antimuscarinic potency and bladder selectivity of PNU-200577, a major metabolite of tolterodine. Pharmacol Toxicol. 1997 Oct;81(4):169-72. [Content Brief]

5-Hydroxymethyl tolterodine formate Related Classifications

Neurological Disease

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Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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5-Hydroxymethyl tolterodine formate380636-49-7PNU-200577PNU200577PNU 200577mAChRMuscarinic acetylcholine receptorInhibitorinhibitorinhibit

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5-Hydroxymethyl tolterodine formate (Synonyms: PNU-200577 formic)

Other Forms of 5-Hydroxymethyl tolterodine formate:

5-Hydroxymethyl tolterodine formate Related Antibodies

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Biological Activity

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References

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