GPR40 agonist 1

Cat. No.: HY-111359: FAQs
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GPR40 agonist 1 is a potent and novel GPR40 full agonist with an EC₅₀ of 2 nM and 17 nM for hGPR40 and rGPR40, respectively.

For research use only. We do not sell to patients.

GPR40 agonist 1 Chemical Structure

CAS No. : 1853982-41-8

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Description	GPR40 agonist 1 is a potent and novel GPR40 full agonist with an EC₅₀ of 2 nM and 17 nM for hGPR40 and rGPR40, respectively.
IC₅₀ & Target	EC50: 2 nM (hGPR40), 17 nM (rGPR40)^[1]
Molecular Weight	479.54
Formula	C₂₇H₃₀FN₃O₄
CAS No.	1853982-41-8
SMILES	COC1=NC=C(F)C(C2=C(CC(C)C)N=C(COC3=CC=CC([C@H](C4CC4)CC(O)=O)=C3)C=N2)=C1
Shipping	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation	Data Sheet (265 KB) Handling Instructions (2659 KB)
References	[1]. Meegalla SK, et al. Discovery of a novel potent GPR40 full agonist. Bioorg Med Chem Lett. 2018 Feb 15;28(4):720-726. [Content Brief]

GPR40 agonist 1 Related Classifications

Metabolic Disease

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Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

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Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPR40 agonist 11853982-41-8Free Fatty Acid ReceptorFFARInhibitorinhibitorinhibit

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GPR40 agonist 1

GPR40 agonist 1 Related Antibodies

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