Rac-Pemafibrate (Synonyms: Rac-K13675)

Cat. No.: HY-17618A: FAQs
Data Sheet Handling Instructions

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Pemafibrate racemate (K13675 racemate) is the racemate of pemafibrate, and activates PPARα activity, with EC₅₀s of 1 nM, >10 μM and 1.7 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively.

For research use only. We do not sell to patients.

Rac-Pemafibrate Chemical Structure

CAS No. : 848258-31-1

Size	Price	Stock
5 mg	USD 80	Ask For Quote & Lead Time
10 mg	USD 130	Ask For Quote & Lead Time
25 mg	USD 250	Ask For Quote & Lead Time
50 mg	USD 400	Ask For Quote & Lead Time
100 mg	USD 680	Ask For Quote & Lead Time

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This product is a controlled substance and not for sale in your territory.

Other Forms of Rac-Pemafibrate:

Pemafibrate In-stock
Pemafibrate-d₄ Get quote

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PPARα PPARβ/δ PPARγ PPAR PPARδ

Biological Activity
Purity & Documentation
References
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Description

IC₅₀ & Target^[1]

h-PPARα

1 nM (EC₅₀)

h-PPARδ

1.7 μM (EC₅₀)

In Vitro

Pemafibrate racemate activates PPARα activity, with EC₅₀s of 1 nM, >10 μM and 1.7 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

490.55

Formula

C₂₈H₃₀N₂O₆

CAS No.

848258-31-1

SMILES

CCC(OC1=CC=CC(CN(C2=NC3=CC=CC=C3O2)CCCOC4=CC=C(OC)C=C4)=C1)C(O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Yamazaki Y, et al. Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor alpha agonists. Bioorg Med Chem Lett. 2007 Aug 15;17(16):4689-93. Epub2007 May 24. [Content Brief]

Rac-Pemafibrate Related Classifications

Inflammation/Immunology

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Rac-Pemafibrate848258-31-1Rac-K13675PPARPeroxisome proliferator-activated receptorsInhibitorinhibitorinhibit

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