2. Signaling Pathways
  3. Epigenetics
  4. Histone Methyltransferase
  5. SMYD2 Isoform
  6. SMYD2 Inhibitor

SMYD2 Inhibitor

SMYD2 Inhibitors (5):

Cat. No. Product Name Effect Purity
  • HY-15226
    AZ505
    		Inhibitor 99.99%
    AZ505 is a potent and selective SMYD2 inhibitor with an IC50 of 0.12 μM.
  • HY-19313
    LLY-507
    		Inhibitor 98.28%
    LLY-507 is a potent and selective inhibitor of protein-lysine methyltransferase SMYD2. LLY-507 potently inhibits the ability of SMYD2 to methylate p53 peptide with an IC50 <15 nM. LLY-507 serves as a valuable chemical probe to aid in the dissection of SMYD2 function in cancer and other biological processes.
  • HY-19546
    BAY-598
    		Inhibitor 99.30%
    BAY-598 is selective small molecule inhibitor of SMYD2 with an IC50 of 27 nM.
  • HY-134828
    AZ506
    		Inhibitor 99.74%
    AZ506 is a potent SMYD2 inhibitor with an IC50 of 17 nM. AZ506 inhibits SMYD2 methyltransferase activity in cells, leading to a decrease in the SMYD2-mediated methylation signal.
  • HY-19563
    A-893
    		Inhibitor
    A-893 is a cell-active inhibitor of Methyltransferase SMYD2, with an IC50 of 2.8 nM.