1. Signaling Pathways
  2. GPCR/G Protein
  3. GPR52
  4. GPR52 Antagonist

GPR52 Antagonist

GPR52 Antagonist (1):

Cat. No. Product Name Effect Purity
  • HY-145468
    GPR52 antagonist-1
    Antagonist 99.80%
    GPR52 antagonist-1 (Compound 43) is a GPR52 antagonist with an IC50 of 0.63 μM. GPR52 antagonist-1 reduces mHTT (mutant huntingtin protein) levels by targeting GPR52 and promotes survival of mouse primary striatal neurons.