2. Signaling Pathways
  3. GPCR/G Protein
  4. Neuromedin U Receptor (NMUR)
  5. Neuromedin U Receptor (NMUR) Antagonist

Neuromedin U Receptor (NMUR) Antagonist

Neuromedin U Receptor (NMUR) Isoform Comparison

Neuromedin U Receptor (NMUR) Antagonists (3):

Cat. No. Product Name Effect Purity
  • HY-145086
    R-PSOP
    		Antagonist 99.90%
    R-PSOP is highly potent and selective nonpeptidic NMUR2 antagonist. R-PSOP binds to NMUR2 with the Kis of 52 and 32 nM for the human and rat NMUR2, respectively. R-PSOP shows moderate CNS penetration. R-PSOP can be used for the research of the eating disorders, obesity, pain, and stress-related disorders.
  • HY-P10473A
    CPN-351 TFA
    		Antagonist
    CPN-351 TFA (compound 9a), a pentapeptide, is a selective antagonist of human NMUR1 with a pA2 of 7.35. The antagonistic effect of CPN-351 TFA on human NMUR1 is 10 times higher than that on NMUR2. CPN-351 TFA can be used in the study of inflammation. X
  • HY-P10473
    CPN-351
    		Antagonist
    CPN-351 (compound 9a), a pentapeptide, is a selective antagonist of human NMUR1 with a pA2 of 7.35. The antagonistic effect of CPN-351 on human NMUR1 is 10 times higher than that on NMUR2. CPN-351 can be used in the study of inflammation.