2. GPCR/G Protein
  3. Adenosine Receptor
  4. A1AR antagonist 6

A1AR antagonist 6 (compound 15) is a potent and selective A1AR (A1 adenosine receptor) antagonist, with a pIC50 of 6.38 and a pKi of 7.13.

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A1AR antagonist 6 Chemical Structure

A1AR antagonist 6 Chemical Structure

CAS No. : 329693-22-3

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A1AR antagonist 6 Related Antibodies

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Description

A1AR antagonist 6 (compound 15) is a potent and selective A1AR (A1 adenosine receptor) antagonist, with a pIC50 of 6.38 and a pKi of 7.13[1].

IC50 & Target

hA1AR

7.13 (pKi)

hA2AAR

<4 (pKi)

Molecular Weight

293.32

Formula

C17H15N3O2
CAS No.
SMILES

N#CC1=C(N=C2CCCCC2=C1C3=CC=C4OCOC4=C3)N
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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A1AR antagonist 6 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

A1AR antagonist 6329693-22-3Adenosine ReceptorP1 receptorA1 adenosine receptorAntagonistInhibitorinhibitorinhibit

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