2. GPCR/G Protein
  3. Angiotensin Receptor
  4. AT1R antagonist 2

AT1R antagonist 2 (compound 6) is a potent AT1R selective ligand. AT1R antagonist 2 exhibits a fair AT1R affinity, with a Ki of 26 nM.

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AT1R antagonist 2 Chemical Structure

AT1R antagonist 2 Chemical Structure

CAS No. : 2848719-76-4

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AT1R antagonist 2 Related Antibodies

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Description

AT1R antagonist 2 (compound 6) is a potent AT1R selective ligand. AT1R antagonist 2 exhibits a fair AT1R affinity, with a Ki of 26 nM[1].

IC50 & Target

Ki: 26 nM (AT1R), 480 nM (AT2R)[1]
Molecular Weight

583.77

Formula

C29H37N5O4S2
CAS No.
SMILES

CCCCOC(NS(=O)(C1=C(N=C(S1)CC(C)C)C2=CC=C(C=C2)CN3C(CC)=NC4=C3N=C(C=C4C)C)=O)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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AT1R antagonist 2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

AT1R antagonist 22848719-76-4Angiotensin Receptorphenylthiazole derivativeHEK-293 cellsphenylthiazole scaffoldphenylthiazole carbamatesAngiotensin II type 2 receptorInhibitorinhibitorinhibit

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AT1R antagonist 2
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HY-146436
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