2. GPCR/G Protein Neuronal Signaling
  3. GPR119
  4. BMS-986034

BMS-986034 is an orally active ingredient (API) that is an agonist of GPR119..

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BMS-986034 Chemical Structure

BMS-986034 Chemical Structure

CAS No. : 1492631-88-5

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BMS-986034 Related Antibodies

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Description

BMS-986034 is an orally active ingredient (API) that is an agonist of GPR119.[1].

IC50 & Target

GPR119[1]
Cellular Effect
Cell Line Type Value Description References
HEK293 EC50
3 nM
Compound: 4
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
[PMID: 24900860]
Molecular Weight

531.39

Formula

C24H24Cl2N6O4
CAS No.
SMILES

O=C1C=C(C(Cl)=CN1C2=NC(C)=C(C=C2)N3C([C@@H](CC3)O)=O)OC4CCN(CC4)C5=NC=C(C=N5)Cl
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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BMS-986034 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

BMS-9860341492631-88-5BMS986034BMS 986034GPR119G Protein-Coupled Receptor 119Inhibitorinhibitorinhibit

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