2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation Membrane Transporter/Ion Channel
  3. Histamine Receptor mAChR Potassium Channel Sodium Channel Calcium Channel
  4. Brompheniramine maleate (Standard)

Brompheniramine maleate (Standard) 

Cat. No.: HY-B0480R Purity: ≥98%
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Brompheniramine (maleate) (Standard) is the analytical standard of Brompheniramine (maleate). This product is intended for research and analytical applications. Brompheniramine ((±)-Brompheniramine) maleate is a potent and orally active antihistamine of the alkylamine class. Brompheniramine maleate is a selective histamine H1 receptor antagonist with a Kd of 6.06 nM. Brompheniramine maleate can block the hERG channels, calcium channels, and sodium channels with IC50s of 0.90 μM, 16.12 μM and 21.26 μM, respectively. Brompheniramine maleate has anticholinergic, antidepressant and anesthetic properties and can be used for allergic rhinitis research.

For research use only. We do not sell to patients.

Brompheniramine maleate (Standard) Chemical Structure

Brompheniramine maleate (Standard) Chemical Structure

CAS No. : 980-71-2

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Description

Brompheniramine (maleate) (Standard) is the analytical standard of Brompheniramine (maleate). This product is intended for research and analytical applications. Brompheniramine ((±)-Brompheniramine) maleate is a potent and orally active antihistamine of the alkylamine class. Brompheniramine maleate is a selective histamine H1 receptor antagonist with a Kd of 6.06 nM. Brompheniramine maleate can block the hERG channels, calcium channels, and sodium channels with IC50s of 0.90 μM, 16.12 μM and 21.26 μM, respectively. Brompheniramine maleate has anticholinergic, antidepressant and anesthetic properties and can be used for allergic rhinitis research.

Molecular Weight

435.31

Formula

C20H23BrN2O4
CAS No.
SMILES

O=C(O)/C=C\C(O)=O.CN(C)CCC(C1=CC=CC=N1)C2=CC=C(Br)C=C2
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
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Brompheniramine maleate (Standard) Related Classifications

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Keywords:

Brompheniramine maleate (Standard)980-71-2Histamine ReceptormAChRPotassium ChannelSodium ChannelCalcium ChannelMuscarinic acetylcholine receptorKcsANa channelsNa+ channelsCa2+ channelsCa channelsanticholinergicantidepressantsedativecommon coldallergic rhinitisantihistamineInhibitorinhibitorinhibit

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