1. Stem Cell/Wnt TGF-beta/Smad Metabolic Enzyme/Protease
  2. PKA Phosphodiesterase (PDE)
  3. 209783-80-2

209783-80-2

Entinostat Chemical Structure

209783-80-2

Chemical Structure

  • Entinostat
  • Synonym(s): MS-275; SNDX-275
  • CAS No: 209783-80-2
    Formula: C21H20N4O3
    Molecular Weight: 376.41
  • IUPAC Name: pyridin-3-ylmethyl (4-((2-aminophenyl)carbamoyl)benzyl)carbamate
  • InChIKey: INVTYAOGFAGBOE-UHFFFAOYSA-N
  • SMILES: O=C(NCC1=CC=C(C=C1)C(NC2=CC=CC=C2N)=O)OCC3=CC=CN=C3

Biological Activity: Entinostat is an oral and selective class I HDAC inhibitor, with IC50s of 243 nM, 453 nM, and 248 nM for HDAC1, HDAC2, and HDAC3, respectively.

Cat. No. Product Name Purity Description
HY-12163 Entinostat 99.82% Entinostat is an oral and selective class I HDAC inhibitor, with IC50s of 243 nM, 453 nM, and 248 nM for HDAC1, HDAC2, and HDAC3, respectively.
HY-12163S Entinostat-d4 Entinostat-d4 is the deuterium labeled Entinostat. Entinostat is an oral and selective class I HDAC inhibitor, with IC50s of 243 nM, 453 nM, and 248 nM for HDAC1, HDAC2, and HDAC3, respectively.