2. MAPK/ERK Pathway Cell Cycle/DNA Damage
  3. Ribosomal S6 Kinase (RSK) YB-1
  4. 2765539-92-0

2765539-92-0

(S,R)-LSN3318839 Chemical Structure

2765539-92-0

Chemical Structure

  • (S,R)-LSN3318839
  • CAS No: 2765539-92-0
    Formula: C26H23Cl2N3O2
    Molecular Weight: 480.39
  • InChIKey: JPJWHCNGSBCZMI-LSDHHAIUSA-N
  • SMILES: C[C@@H](C1=CC=CC=C1C2=NC=C3N=CN(C3=C2)[C@@H](C4=C(C(C5CC5)=CC=C4Cl)Cl)C)C(O)=O

Biological Activity: (S,R)-LSN3318839 is the stereoisomer of LSN3318839 (HY-142162). LSN3318839 is an orally active positive modulator of the glucagon-like peptide-1 receptor (GLP-1R). LSN3318839 can increase the secretion of insulin and has the effect of lowering blood sugar[1].

Cat. No. Product Name Purity Description
HY-140171 m-PEG5-sulfonic acid m-PEG5-sulfonic acid is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs.

References

[1]. Willard FS, et al., Discovery of an Orally Efficacious Positive Allosteric Modulator of the Glucagon-like Peptide-1 Receptor. J Med Chem. 2021 Mar 25;64(6):3439-3448. [Content Brief]

Keywords:

(S,R)-LSN3318839