2. Membrane Transporter/Ion Channel
  3. OAT
  4. 53818-10-3

53818-10-3

4’-Hydroxy Trazodone Chemical Structure

53818-10-3

Chemical Structure

  • 4’-Hydroxy Trazodone
  • CAS No: 53818-10-3
    Molecular Weight: 387.86
  • IUPAC Name: 2-(3-(4-(3-chloro-4-hydroxyphenyl)piperazin-1-yl)propyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
  • InChIKey: FNUZSRSXQFIOPL-UHFFFAOYSA-N
  • SMILES: ClC1=CC(N2CCN(CCCN3N=C(C=CC=C4)N4C3=O)CC2)=CC=C1O

Biological Activity: 4’-hydroxy Trazodone is a metabolite of the antidepressant and sedative trazodone. It is an inhibitor of organic anion transporter 3 (OAT3; Ki=16.9 μM) and is selective for OAT3 over OAT1 (Ki=>200 μM).

Cat. No. Product Name Purity Description
HY-W740244 4’-Hydroxy Trazodone 4’-hydroxy Trazodone is a metabolite of the antidepressant and sedative trazodone. It is an inhibitor of organic anion transporter 3 (OAT3; Ki=16.9 μM) and is selective for OAT3 over OAT1 (Ki=>200 μM).

Keywords:

4’-Hydroxy Trazodone