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  6. 57775-22-1

57775-22-1

Etoperidone hydrochloride Chemical Structure

57775-22-1

Chemical Structure

  • Etoperidone hydrochloride
  • CAS No: 57775-22-1
    Formula: C19H29Cl2N5O
    Molecular Weight: 414.37
  • IUPAC Name: 2-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-4,5-diethyl-2,4-dihydro-3H-1,2,4-triazol-3-one hydrochloride
  • InChIKey: BHKPQZVLIZKSAG-UHFFFAOYSA-N
  • SMILES: O=C1N(CCCN2CCN(CC2)C3=CC(Cl)=CC=C3)N=C(CC)N1CC.Cl

Biological Activity: Etoperidone hydrochloride, an antidepressant agent, is an orally active serotonin and nor-adrenaline re-uptake antagonist. Etoperidone hydrochloride shows Kd values of 36 nM, 38 nM, 85 nM, and 570 nM for 5-HT2 receptor, α1-adrenergic receptor, 5-HT1A receptor, and α2-adrenergic receptor, respectively[1][2].

Cat. No. Product Name Purity Description
HY-106617A Etoperidone hydrochloride Etoperidone hydrochloride, an antidepressant agent, is an orally active serotonin and nor-adrenaline re-uptake antagonist. Etoperidone hydrochloride shows Kd values of 36 nM, 38 nM, 85 nM, and 570 nM for 5-HT2 receptor, α1-adrenergic receptor, 5-HT1A receptor, and α2-adrenergic receptor, respectively.
HY-106617AS Etoperidone-d8 hydrochloride Etoperidone-d8 (hydrochloride) is the deuterium labeled Etoperidone hydrochloride.

References

[1]. B Cusack, et al. Binding of antidepressants to human brain receptors: focus on newer generation compounds. Psychopharmacology (Berl). 1994 May;114(4):559-65. [Content Brief]
[2]. G W Caldwell, et al. Evaluation of the absorption, excretion and metabolism of [14C] etoperidone in man. Xenobiotica. 2001 Nov;31(11):823-39. [Content Brief]

Keywords:

Etoperidone hydrochlorideEtoperidone-d8 hydrochloride