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CASK-IN-1 is a highly potent and selective CASK inhibitor with a Kd value of 0.022 μM.

For research use only. We do not sell to patients.

CASK-IN-1 Chemical Structure

CASK-IN-1 Chemical Structure

CAS No. : 2755241-73-5

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CASK-IN-1 Related Antibodies

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Description

CASK-IN-1 is a highly potent and selective CASK inhibitor with a Kd value of 0.022 μM.

Molecular Weight

610.34

Formula

C24H30Br2N6O3
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(C1=CN=C(N=C1NC2CCCC2)NCC3=CC(Br)=C(C=C3Br)C)NCCCN4CCOC4=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 12.21 mg/mL (20.01 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.6384 mL 8.1922 mL 16.3843 mL
5 mM 0.3277 mL 1.6384 mL 3.2769 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

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Volume (start)

V1

=
Concentration (final)

C2

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Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 1.6384 mL 8.1922 mL 16.3843 mL 40.9608 mL
5 mM 0.3277 mL 1.6384 mL 3.2769 mL 8.1922 mL
10 mM 0.1638 mL 0.8192 mL 1.6384 mL 4.0961 mL
15 mM 0.1092 mL 0.5461 mL 1.0923 mL 2.7307 mL
20 mM 0.0819 mL 0.4096 mL 0.8192 mL 2.0480 mL
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CASK-IN-1 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CASK-IN-12755241-73-5OthersInhibitorinhibitorinhibit

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CASK-IN-1
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HY-115719
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