2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. Calcium Channel
  4. Cav 2.2/3.2 blocker 1

Cav 2.2/3.2 blocker 1 (Compound 9e) is a neuronal calcium channel blocker with IC50 values of 78 μM and 80 μM against Cav2.2 and Cav3.2, respectively. Cav 2.2/3.2 blocker 1 can penetrate the CNS.

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Cav 2.2/3.2 blocker 1 Chemical Structure

Cav 2.2/3.2 blocker 1 Chemical Structure

CAS No. : 2987640-67-3

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Cav 2.2/3.2 blocker 1 Related Antibodies

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N-type calcium channel L-type calcium channel P/Q-type calcium channel T-type calcium channel Calcium Channel

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Description

Cav 2.2/3.2 blocker 1 (Compound 9e) is a neuronal calcium channel blocker with IC50 values of 78 μM and 80 μM against Cav2.2 and Cav3.2, respectively. Cav 2.2/3.2 blocker 1 can penetrate the CNS[1].

IC50 & Target

Cav3.2

80 μM (IC50)

CaV2.2

78 μM (IC50)

Molecular Weight

442.55

Formula

C28H30N2O3
CAS No.
SMILES

O=C(N1C2=CC=CC=C2CCC3=CC=CC=C31)C4=CC=C(OCCCN5CCOCC5)C=C4
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Cav 2.2/3.2 blocker 1 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Cav 2.2/3.2 blocker 12987640-67-3Calcium ChannelCa2+ channelsCa channelsCNS penetrabilityN-type calcium channelCav2.2Cav3.2T-type calcium channelInhibitorinhibitorinhibit

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