2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. CB1 antagonist 5

CB1 antagonist 5 (Compound 25) is an antagonist for CB1 cannabinoid receptor, with a Ki of 243 nM and an EC50 of 195 nM.

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CB1 antagonist 5 Chemical Structure

CB1 antagonist 5 Chemical Structure

CAS No. : 878533-35-8

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CB1 antagonist 5 Related Antibodies

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Description

CB1 antagonist 5 (Compound 25) is an antagonist for CB1 cannabinoid receptor, with a Ki of 243 nM and an EC50 of 195 nM[1].

IC50 & Target

hCB1

195 nM (EC50)

hCB1

243 nM (Ki)

Molecular Weight

486.16

Formula

C21H14Br2N2O2
CAS No.
SMILES

O=C1N(C(C(N1C2=CC=C(C=C2)Br)C3=CC=CC=C3)=O)C4=CC=C(C=C4)Br
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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CB1 antagonist 5 Related Classifications

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CB1 antagonist 5878533-35-8Cannabinoid ReceptorInhibitorinhibitorinhibit

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