1. GPCR/G Protein Neuronal Signaling
  2. Cannabinoid Receptor
  3. CB1 antagonist 5

CB1 antagonist 5 (Compound 25) is an antagonist for CB1 cannabinoid receptor, with a Ki of 243 nM and an EC50 of 195 nM.

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CB1 antagonist 5 Chemical Structure

CB1 antagonist 5 Chemical Structure

CAS No. : 878533-35-8

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Description

CB1 antagonist 5 (Compound 25) is an antagonist for CB1 cannabinoid receptor, with a Ki of 243 nM and an EC50 of 195 nM[1].

IC50 & Target

hCB1

195 nM (EC50)

hCB1

243 nM (Ki)

Molecular Weight

486.16

Formula

C21H14Br2N2O2

CAS No.
SMILES

O=C1N(C(C(N1C2=CC=C(C=C2)Br)C3=CC=CC=C3)=O)C4=CC=C(C=C4)Br

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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CB1 antagonist 5
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HY-120653
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