2. Epigenetics
  3. Histone Acetyltransferase
  4. CBP/p300-IN-16

CBP/p300-IN-16 (compound 1) is a potent EP300/CBP HAT inhibitor with IC50s of 0.61, 2.24 µM for HAT EP300 and LK2 H3K27, respectively.

For research use only. We do not sell to patients.

CBP/p300-IN-16 Chemical Structure

CBP/p300-IN-16 Chemical Structure

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CBP/p300-IN-16 Related Antibodies

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Description

CBP/p300-IN-16 (compound 1) is a potent EP300/CBP HAT inhibitor with IC50s of 0.61, 2.24 µM for HAT EP300 and LK2 H3K27, respectively[1].

IC50 & Target[1]

LK2 H3K27

2.24 μM (IC50)

Molecular Weight

449.54

Formula

C26H31N3O4
SMILES

O=C(N1CCOC[C@H](CC2=CC=CC3=C2C=NN3)C1)C4(C5=CC=C(OC)C=C5)CCOCC4
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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CBP/p300-IN-16 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CBP/p300-IN-16Histone AcetyltransferaseHATsHATanticancerhistone acetyltransferasesInhibitorinhibitorinhibit

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