2. Epigenetics
  3. Histone Acetyltransferase
  4. CBP/p300-IN-17

CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively.

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CBP/p300-IN-17 Chemical Structure

CBP/p300-IN-17 Chemical Structure

CAS No. : 2259640-87-2

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CBP/p300-IN-17 Related Antibodies

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Description

CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively[1].

IC50 & Target[1]

EP300

.18 μM (IC50)

LK2 H3K27

0.69 μM (IC50)

Molecular Weight

432.51

Formula

C25H28N4O3
CAS No.
SMILES

O=C([C@@H]1N(C(C2(C3=CC=C(OC)C=C3)CCCC2)=O)CCC1)NC4=CC=CC5=C4C=NN5
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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CBP/p300-IN-17 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CBP/p300-IN-172259640-87-2Histone AcetyltransferaseHATsHATanticancerhistone acetyltransferasesInhibitorinhibitorinhibit

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