2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor Dopamine Receptor
  4. Cinitapride monotartrate

Cinitapride monotartrate is a 5-HT1A and 5-HT4 agonist. Cinitapride monotartrate is also a 5-HT2A and D2 antagonist. Cinitapride monotartrate can be used for the research of functional dyspepsia.

For research use only. We do not sell to patients.

Cinitapride monotartrate Chemical Structure

Cinitapride monotartrate Chemical Structure

CAS No. : 1207859-16-2

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Based on 1 publication(s) in Google Scholar

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Cinitapride monotartrate Related Antibodies

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Description

Cinitapride monotartrate is a 5-HT1A and 5-HT4 agonist. Cinitapride monotartrate is also a 5-HT2A and D2 antagonist. Cinitapride monotartrate can be used for the research of functional dyspepsia[1][2].

IC50 & Target[1]

5-HT2 Receptor

 

5-HT1 Receptor

 

5-HT4 Receptor

 

D2 Receptor

 

In Vivo

Cinitapride (intraperitoneal injection; 0.25-1 mg/kg; once) shows gastroprotective effetcs in gastric ulceration rat model[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male Wistar rats with gastric ulceration[2]
Dosage: 0.25-1 mg/kg
Administration: Intraperitoneal injection; 0.25-1 mg/kg; once
Result: Reduced haemorrhagic lesions compared with the ulcerated control group.
Decreased the percentage of ulceration to 28.76% at the highest dose (1 mg/kg).
Attenuated the increase myeloperoxidase activity (p<0.05, p<0.01).
Increased GSH-px activity in the gastric mucosa.
Molecular Weight

552.57

Formula

C25H36N4O10
CAS No.
SMILES

O=C(NC1CCN(CC2CC=CCC2)CC1)C3=CC([N+]([O-])=O)=C(N)C=C3OCC.O=C(O)[C@H](O)[C@@H](O)C(O)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Cinitapride monotartrate Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Cinitapride monotartrate1207859-16-25-HT ReceptorDopamine ReceptorSerotonin Receptor5-hydroxytryptamine Receptorfunctional dyspepsiawell tolerateddelayed gastric emptyingInhibitorinhibitorinhibit

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