2. GPCR/G Protein Neuronal Signaling
  3. Dopamine Receptor
  4. D3R ligand 1

D3R ligand 1 (compound 23b) is a potent and selective ligand of dopamine receptor D3R (Ki=66 nM), containing a THPB template. D3R ligand 1 is also an antagonist for both G-protein- and β-arrestin-based signaling.

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D3R ligand 1 Chemical Structure

D3R ligand 1 Chemical Structure

CAS No. : 2983777-91-7

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D3R ligand 1 Related Antibodies

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Description

D3R ligand 1 (compound 23b) is a potent and selective ligand of dopamine receptor D3R (Ki=66 nM), containing a THPB template. D3R ligand 1 is also an antagonist for both G-protein- and β-arrestin-based signaling[1].

IC50 & Target

D3 Receptor

66 nM (Ki)

Molecular Weight

455.59

Formula

C27H37NO5
CAS No.
SMILES

OC1=C(C=C(C2=C1)CCN3[C@H]2CC4=CC=C(C(OCCOCC)=C4C3)O)OCCCCCC
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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D3R ligand 1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

D3R ligand 12983777-91-7Dopamine ReceptorInhibitorinhibitorinhibit

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