1. GPCR/G Protein Neuronal Signaling
  2. Dopamine Receptor
  3. D4R antagonist-2

D4R antagonist-2 (compound 33) is a D4R antagonist. D4R antagonist-2 has a IC50 value of 210 nM, and a Ki value of 59 nM for D4R. D4R antagonist-2 can be used in the Parkinson's disease research.

For research use only. We do not sell to patients.

D4R antagonist-2 Chemical Structure

D4R antagonist-2 Chemical Structure

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Description

D4R antagonist-2 (compound 33) is a D4R antagonist. D4R antagonist-2 has a IC50 value of 210 nM, and a Ki value of 59 nM for D4R. D4R antagonist-2 can be used in the Parkinson's disease research[1].

IC50 & Target

D4 Receptor

 

Molecular Weight

391.48

Formula

C24H26FN3O

SMILES

O=C(N1CC2(CCN(CC3=CNC4=C3C=CC(F)=C4)CC2)C1)C5=CC=CC=C5C

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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D4R antagonist-2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
D4R antagonist-2
Cat. No.:
HY-163703
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