2. Metabolic Enzyme/Protease Neuronal Signaling GPCR/G Protein Membrane Transporter/Ion Channel
  3. Dipeptidyl Peptidase GPR119 Potassium Channel
  4. DPP-4/GPR119 modulator 1

DPP-4/GPR119 modulator 1 (Compound 22) is an orally active dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist. DPP-4/GPR119 modulator 1 shows blood glucose-lowering effect and moderate inhibition on hERG channel with an IC50 of 4.9 μM. DPP-4/GPR119 modulator 1 can be used for diabetes research. DPP-4/GPR119 modulator 1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

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DPP-4/GPR119 modulator 1 Chemical Structure

DPP-4/GPR119 modulator 1 Chemical Structure

CAS No. : 2411099-68-6

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DPP-4/GPR119 modulator 1 Related Antibodies

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Description

DPP-4/GPR119 modulator 1 (Compound 22) is an orally active dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist. DPP-4/GPR119 modulator 1 shows blood glucose-lowering effect and moderate inhibition on hERG channel with an IC50 of 4.9 μM. DPP-4/GPR119 modulator 1 can be used for diabetes research[1][1]. DPP-4/GPR119 modulator 1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

IC50 & Target

DPP-4

 

Molecular Weight

623.15

Formula

C30H39ClN10O3
CAS No.
SMILES

CC#CCN1C(N2CCC[C@H](C2)N)=NC3=C1C(N(C(N3C)=O)CCCN4CCN(CC4)C5=NC(C6=CC=CC=C6)=NO5)=O.Cl
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Room temperature in continental US; may vary elsewhere.
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Purity & Documentation
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DPP-4/GPR119 modulator 1 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

DPP-4/GPR119 modulator 12411099-68-6Dipeptidyl PeptidaseGPR119Potassium ChannelDPPG Protein-Coupled Receptor 119KcsAICR miceKKAy miceglucose-lowering effectorally activediabetesInhibitorinhibitorinhibit

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