2. PROTAC
  3. E3 Ligase Ligand-Linker Conjugates
  4. E3 ligase Ligand-Linker Conjugate 39

E3 ligase Ligand-Linker Conjugate 39 is a conjugate of E3 ligase ligand and linker, consisting of Thalidomide (HY-14658) and the corresponding Linker. E3 ligase Ligand-Linker Conjugate 39 can serve as a Cereblon ligand to recruit CRBN protein and serve as a key intermediate for the synthesis of complete PROTAC molecules.

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E3 ligase Ligand-Linker Conjugate 39 Chemical Structure

E3 ligase Ligand-Linker Conjugate 39 Chemical Structure

CAS No. : 2632308-04-2

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E3 ligase Ligand-Linker Conjugate 39 Related Antibodies

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View All E3 Ligase Ligand-Linker Conjugates Isoform Specific Products:

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von Hippel-Lindau (VHL) MDM2 Cereblon cIAP1 Aryl Hydrocarbon Receptor

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Description

E3 ligase Ligand-Linker Conjugate 39 is a conjugate of E3 ligase ligand and linker, consisting of Thalidomide (HY-14658) and the corresponding Linker. E3 ligase Ligand-Linker Conjugate 39 can serve as a Cereblon ligand to recruit CRBN protein and serve as a key intermediate for the synthesis of complete PROTAC molecules.

IC50 & Target

Cereblon (CRBN)[1]
Molecular Weight

497.54

Formula

C25H31N5O6
CAS No.
SMILES

O=C1NC(CCC1N2C(C3=C(C=CC(N4CC(C4)N5CCN(CC5)C(OC(C)(C)C)=O)=C3)C2=O)=O)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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E3 ligase Ligand-Linker Conjugate 39 Related Classifications

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Keywords:

E3 ligase Ligand-Linker Conjugate 392632308-04-2E3 Ligase Ligand-Linker ConjugatesInhibitorinhibitorinhibit

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