2. JAK/STAT Signaling Protein Tyrosine Kinase/RTK Autophagy
  3. EGFR Autophagy
  4. Erlotinib-d6 hydrochloride

Erlotinib-d6 hydrochloride  (Synonyms: CP-358774-d6 hydrochloride; NSC 718781-d6 hydrochloride; OSI-774-d6 hydrochloride)

Cat. No.: HY-12008S Purity: 98.13%
COA Handling Instructions

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Erlotinib-d6 (hydrochloride) a deuterium labeled Erlotinib Hydrochloride. Erlotinib Hydrochloride inhibits purified EGFR kinase with an IC50 of 2 nM[1]. Erlotinib-d6 (hydrochloride) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

For research use only. We do not sell to patients.

Erlotinib-d<sub>6</sub> hydrochloride Chemical Structure

Erlotinib-d6 hydrochloride Chemical Structure

CAS No. : 1189953-78-3

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Based on 1 publication(s) in Google Scholar

Other Forms of Erlotinib-d6 hydrochloride:

Erlotinib-d6 hydrochloride Related Antibodies

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Description

Erlotinib-d6 (hydrochloride) a deuterium labeled Erlotinib Hydrochloride. Erlotinib Hydrochloride inhibits purified EGFR kinase with an IC50 of 2 nM[1]. Erlotinib-d6 (hydrochloride) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

Molecular Weight

435.93

Formula

C22H18D6ClN3O4
CAS No.
Unlabeled CAS

183319-69-9
Appearance

Solid

Color

White to off-white

SMILES

[2H]C([2H])([2H])OCCOC1=CC2=NC=NC(NC3=CC=CC(C#C)=C3)=C2C=C1OCCOC([2H])([2H])[2H].[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

H2O : ≥ 0.1 mg/mL (0.23 mM)

H2O : ≥ 0.1 mg/mL (0.23 mM)

*"≥" means soluble, but saturation unknown.

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Purity & Documentation

Purity: 98.13%

COA (251 KB)

Handling Instructions (2659 KB)
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Erlotinib-d6 hydrochloride Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Erlotinib-d61189953-78-3CP-358774-d6NSC 718781-d6OSI-774-d6EGFRAutophagyEpidermal growth factor receptorErbB-1HER1Inhibitorinhibitorinhibit

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