2. GPCR/G Protein
  3. Free Fatty Acid Receptor
  4. FFA2 agonist-1

FFA2 agonist-1 (Compound 4) is the agonist for Free fatty acid receptor 2 (FFA2/GPR43) with an EC50 of 81 nM. FFA2 agonist-1 exhibits activity in β-arrestin-2 recruitment assay and cAMP inhibition assay with EC50 of 1.2 μM and 0.53 μM. FFA2 agonist-1 leads to appetite regulating peptide YY (PYY) mucosal responses, inhibits the fat accumulation, intestinal functions and food intake, and can be used for obesity research.

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FFA2 agonist-1 Chemical Structure

FFA2 agonist-1 Chemical Structure

CAS No. : 1312799-06-6

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FFA2 agonist-1 Related Antibodies

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Description

FFA2 agonist-1 (Compound 4) is the agonist for Free fatty acid receptor 2 (FFA2/GPR43) with an EC50 of 81 nM. FFA2 agonist-1 exhibits activity in β-arrestin-2 recruitment assay and cAMP inhibition assay with EC50 of 1.2 μM and 0.53 μM. FFA2 agonist-1 leads to appetite regulating peptide YY (PYY) mucosal responses, inhibits the fat accumulation, intestinal functions and food intake, and can be used for obesity research[1].

IC50 & Target

EC50: 81 nM (FFA2/GPR43)
Molecular Weight

435.90

Formula

C25H22ClNO4
CAS No.
SMILES

O=C(C1=CC=C(C2=C(C=CC=C2)OC)C=C1)N3[C@@H](C4=C(C=CC=C4)Cl)CC[C@H]3C(O)=O
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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FFA2 agonist-1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

FFA2 agonist-11312799-06-6Free Fatty Acid ReceptorFFARobesityPPYappetite regulatingInhibitorinhibitorinhibit

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